ACTIVE – Cyclobenzaprine Kit

NDC #: 45861-0103-01

ACTIVE Cyclobenzaprine Kit facilitates customized in-house compounding by packaging pre-weighed Cyclobenzaprine 5% together with Alba-Derm, an emollient base with excellent penetration. When used topically at the site of pain, Cyclobenzaprine effectively relaxes muscle tissue and delivers an analgesic effect with minimal systemic absorption, making it especially beneficial for elderly patients and those with can’t tolerate oral muscle relaxants.

Pharmaceutica North America is proud to provide our ACTIVE Cyclobenzaprine Kit because it offers a convenient way for clinicians to efficiently prepare topical treatment for in-house patients. Like all of our products, the active ingredients in this kit are manufactured and distributed in accordance with cGMP at an FDA and DEA registered facility.

Approved and Potential Uses of Topical Cyclobenzaprine:

Cyclobenzaprine is a skeletal muscle relaxant that’s structurally related to tricyclic antidepressants. When applied topically, Cyclobenzaprine relieves pain and spasms associated with musculoskeletal conditions through various mechanisms, including blocking uptake of norepinephrine and serotonin, interactions with mu-opioid receptors and sodium channels, and potent peripheral anticholinergic effects.

Alba-Derm is an oil-in-water emulsion specially formulated to provide a highly penetrating delivery vehicle for a wide range of active pharmaceutical ingredients. As a superior emollient that’s paraben-free, Alba-Derm is recommended for pharmaceutical and cosmetic use.

Consider using ACTIVE Cyclobenzaprine Kit for the following conditions:

  • Muscle spasms – Topical cyclobenzaprine relieves pain and tenderness by relaxing muscle spasms. When used in conjunction with physical therapy, it may improve range of motion.
  • Chronic musculoskeletal conditions – As adjunctive therapy, cyclobenzaprine relieves pain associated with injury to muscles, tendons, ligaments, and joints.
  • Neuropathic pain – Topical application of tricyclic antidepressants helps attenuate nociception, which reduces pain associated with diabetic neuropathy and postherpetic neuralgia.
  • Fibromyalgia and myofascial pain syndrome – When used as adjunctive therapy, topical cyclobenzaprine applied to trigger points may relieve chronic pain.

When you purchase the ACTIVE Cyclobenzaprine Kit from Pharmaceutica North America, you’re guaranteed competitive pricing and stable, high-quality products. Our team of experts stands ready to provide personalized service and ensure a steady supply of the pharmaceuticals you need. Contact us today to learn about our fast shipping and to experience first-class customer service in action.